Patent application number | Description | Published |
20080275235 | NOVEL FUSED HETEROAROMATIC COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS - Novel fused heteroaromatic compounds, including derivatives thereof, to intermediates for their preparation, to pharmaceutical compositions containing them and to their medicinal use are described. The compounds of the present invention are potent inhibitors of transforming growth factor (“TGF”)- | 11-06-2008 |
20090005416 | BENZIMIDAZOLE DERIVATIVES - The present invention relates to a compound of the Formula I | 01-01-2009 |
20090036425 | SUBSTITUTED BICYCLOLACTAM COMPOUNDS - The invention provides compounds of formula (1), | 02-05-2009 |
20090137551 | Substituted Bicyclolactam Compounds - The invention provides compounds of formula (1), | 05-28-2009 |
20100035903 | PYRROLO[2,3-D]PYRIMIDINE COMPOUNDS - A compound of the formula | 02-11-2010 |
20100056571 | NOVEL PYRAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITORS - Novel pyrazole compounds, including derivatives thereof, to intermediates for their preparation, to pharmaceutical compositions containing them and to their medicinal use are described. The compounds of the present invention are potent inhibitors of transforming growth factor (“TGF”)- | 03-04-2010 |
20100197590 | 4-AMINO-7,8-DIHYDROPYRIDO[4,3-d]PYRIMIDIN-5(6H)-ONE DERIVATIVES - The invention provides compounds of Formula (Ia) | 08-05-2010 |
20100197591 | 4-AMINO-7,8-DIHYDROPYRIDO[4,3-d]PYRIMIDIN-5(6H)-ONE DERIVATIVES - The invention provides compounds of the general Formula (I) | 08-05-2010 |
20100204119 | 4-AMINO-5-OXO-7,8-DIHYDROPYRIMIDO[5,4-F][1,4]OXAZEPIN-6(5H)-YL PHENYL DERIVATIVES - The invention provides compounds of Formula (I), | 08-12-2010 |
20100285145 | GPR 119 MODULATORS - Compounds of Formula (I) that modulate the activity of the G-protein-coupled receptor GPR119 and their uses in the treatment of diseases linked to the modulation of the G-protein-coupled receptor GPR119 in animals are described herein. | 11-11-2010 |
20110020460 | GPR 119 MODULATORS - Compounds of Formula I that modulate the activity of the G-protein-coupled receptor GPR119 and their uses in the treatment of diseases linked to the modulation of the G-protein-coupled receptor GPR119 in animals are described herein. | 01-27-2011 |
20120157495 | BENZIMIDAZOLE DERIVATIVES - The present invention relates to a compound of the Formula I | 06-21-2012 |
20120295845 | IMIDAZO-PYRAZOLES AS GPR119 INHIBITORS - Compounds of formula (I) wherein: X is (A) or (B); Y is O or a bond; R | 11-22-2012 |
20130072427 | GPR 119 MODULATORS - Compounds of formula (I) that modulate the activity of the G-protein-coupled receptor GPR119 and their uses in the treatment of diseases linked to the modulation of the G-protein-coupled receptor GPR119 in animals are described herein. | 03-21-2013 |