Patent application number | Description | Published |
20080234266 | Squaric Acid Derivatives II -
Compounds of the formula (I), in which R, X, X′ and R | 09-25-2008 |
20080306042 | Triazole Derivatives - Novel triazole derivatives are inhibitors of TGF-beta receptor I kinase, and can be employed, inter alia, for the treatment of tumours. | 12-11-2008 |
20080312244 | Squaric Acid Derivatives as Protein Kinase Inhibitors - Compounds of the formula I, in which R, X, R | 12-18-2008 |
20080318934 | Diazepinoes - The invention relates to compounds of the formula (I), to the preparation and use thereof for the preparation of a medicament for the treatment of diseases, in particular tumours and/or diseases in the development or course of which kinases are involved. | 12-25-2008 |
20090131506 | Oxindoles as Kinase Inhibitors - The present invention relates to oxindoles of the formula I, their use as protein kinase activators or inhibitors, a method for their manufacture, their use for the preparation of a medicament for the treatment of diseases and their use for the manufacture of a pharmaceutical composition. | 05-21-2009 |
20090215799 | HETEROCYCLIC SUBSTITUTED BISARYLUREA DERIVATIVES - The present invention relates to heterocyclic substituted bisarylurea derivatives of formula I, the use of the compounds of formula I as inhibitors of one or more kinases, the use of the compounds of formula I for the manufacture of a pharmaceutical composition and a method of treatment, comprising administering said pharmaceutical composition to a patient. | 08-27-2009 |
20090247584 | PHENOXY-PIPERIDINES FOR THE TREATMENT OF DISEASES SUCH AS SCHIZOPHRENIA AND DEPRESSION - Compounds of the formula (I), in which R | 10-01-2009 |
20100063028 | Triazabenzo[E]Azulene Derivatives for the Treatment Of Tumors - Novel triazabenzo[e]azulene derivatives of the formula, (I) in which R | 03-11-2010 |
20100160356 | NOVEL CYCLOBUTYL COMPOUNDS AS KINASE INHIBITORS - The invention relates to compounds of the formula I, to the preparation and use thereof for the preparation of a medicament for the treatment of diseases, in particular tumours and/or diseases in the formation or course of which protein kinases are involved. | 06-24-2010 |
20100197757 | OXINDOLES AS KINASE INHIBITORS - The present invention relates to oxindoles of the formula I, their use as protein kinase activators or inhibitors, a method for their manufacture, their use for the preparation of a medicament for the treatment of diseases and their use for the manufacture of a pharmaceutical composition. | 08-05-2010 |
20100234369 | 5-CYANOTHIENOPYRIDINES FOR THE TREATMENT OF TUMOURS - Novel 5-cyanothienopyridines of the formula (I), in which R | 09-16-2010 |
20110028472 | THIENOPYRIMIDINES - Novel thienopyrimidines of the formula (I), in which R | 02-03-2011 |
20120101095 | ALKOXY-THIENOPYRIMIDINES AS TGF-BETA RECEPTOR KINASE MODULATORS - Novel alkoxy-thienopyrimidine derivatives of formula (I) | 04-26-2012 |
20130158005 | PYRIMIDINE DERIVATIVES AS FAK INHIBITORS - Compounds of the formula (I), in which R | 06-20-2013 |