Patent application number | Description | Published |
20090163464 | BENZOTHIAZOLE AND BENZOOXAZOLE DERIVATIVES AND METHODS OF USE - Compounds of formula (I) are useful in treating conditions or disorders prevented by or ameliorated by histamine-3 receptor ligands. Also disclosed are pharmaceutical compositions of compounds of formula (I), methods for using such compounds and compositions, and a process for preparing the compounds. | 06-25-2009 |
20090163470 | THIAZOLYLIDINE UREA AND AMIDE DERIVATIVES AND METHODS OF USE THEREOF - The invention relates to novel thiazolylidine urea and amide derivatives that are PAMs of neuronal nicotinic receptors, compositions comprising the same, processes for preparing such compounds, and methods for using such compounds and compositions. | 06-25-2009 |
20090221648 | COMPOSITIONS FOR TREATMENT OF COGNITIVE DISORDERS - The present invention relates to compositions for treatment of cognitive deficits. Such compositions can have a nicotinic acetylcholine receptor ligand, of either α4β2 subtype or α7 nicotinic acetylcholine subtype, and a histamine-3 receptor ligand, a method of using the same, and a related article of manufacture. Combinations of such active agents with psychostimulants or monoamine reuptake inhibitors also is contemplated. | 09-03-2009 |
20100087471 | INDOLE AND INDOLINE DERIVATIVES AND METHODS OF USE THEREOF - The present application relates to indole and indoline derivatives of formula (I), (II), (III), (IV), (V), or (VI) | 04-08-2010 |
20100190776 | Thiazoline and Oxazoline Derivatives and Their Methods of Use - The invention relates to a series of thiazoline and oxazoline derivatives, compositions thereof, and methods of treating conditions and disorders using such compounds. | 07-29-2010 |
20100216748 | Pyrrole Derivatives and Their Methods of Use - The invention relates to a series of substituted pyrrole derivatives, compositions comprising the same, and methods of treating conditions and disorders using such compounds and compositions. | 08-26-2010 |
20100249105 | INDOLE AND INDOLINE DERIVATIVES AND METHODS OF USE THEREOF - The present application relates to indole and indoline derivatives of formula (I), (II), (III), (IV), (V), or (VI) | 09-30-2010 |
20100331294 | 4-SUBSTITUTED-2-AMINO-PYRIMIDINE DERIVATIVES - Compounds of the formula | 12-30-2010 |
20100331353 | 3,9-DIAZASPIRO[5,5]UNDECANE AMIDES AND UREAS AND METHODS OF USE THEREOF - Compounds of formula (I) | 12-30-2010 |
20110098285 | BICYCLIC-SUBSTITUTED AMINES AS HISTAMINE-3 RECEPTOR LIGANDS - Compounds of formula (I) | 04-28-2011 |
20120164070 | BENZOTHIAZOLE AND BENZOOXAZOLE DERIVATIVES AND METHODS OF USE - Compounds of formula (I) | 06-28-2012 |
20120245163 | TRPV1 Antagonists - Disclosed herein are compounds of formula (I) or pharmaceutically acceptable salts, solvates, or combinations thereof, | 09-27-2012 |
20130131036 | NOVEL TRPV3 MODULATORS - Disclosed herein are modulators of TRPV3 of formula (II): | 05-23-2013 |
20130158067 | TRPV1 Antagonists - Disclosed herein are compounds of formula (I): | 06-20-2013 |
20130172334 | TRPV1 ANTAGONISTS - Disclosed herein are compounds of formula (I): | 07-04-2013 |
20140080803 | NOVEL TRPV3 MODULATORS - Disclosed herein are modulators of TRPV3 of Formula (I) | 03-20-2014 |