| Patent application number | Description | Published |
|---|
| 20080200687 | Preparation of Terazole Derivatives - The invention relates to a process for the preparation of (S)-pyrrolidine-1H-tetrazole derivatives of formula | 08-21-2008 |
| 20080207921 | Organic Compounds - The invention related to a novel process, novel process steps and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially renin inhibitors, such as Aliskiren. Inter alia, the invention relates to a process for the manufacture of a compound of the formula III, | 08-28-2008 |
| 20080234490 | Metal Salts of 2' - (1H-Tetrazol-5Yl) -1. 1'-Biphenyl-4-Carboxaldehyde - The invention relates to a method or process for the manufacture of blood pressure lowering agents, such as valsartan, novel intermediates as well as process steps in said synthesis. The method or process leads via the novel intermediate salts of the formula IA, | 09-25-2008 |
| 20080249318 | Process for phenylacetic acid derivatives - A process for the production of a compound of Formula I, or a pharmaceutically acceptable salt thereof, or a pharmaceutically acceptable prodrug ester thereof, | 10-09-2008 |
| 20080262246 | 3-Alkyl-5- (4-Alkyl-5-Oxo-Tetrahydrofutr An -2-Yl) Pyrrolidin-2-One Derivatives As Intermediates In The Synthesis Of Renin Inhibitors - The invention related to a novel process, novel process steps and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially renin inhibitors, such as Aliskiren. Inter alia, the invention relates to a process for the manufacture of a compound of the formula II, | 10-23-2008 |
| 20080312462 | Process for the manufacture of HMG-CoA reductase inhibitory mevalonic acid derivatives - The invention relates to a process for the manufacture of a compound of formula: (Formula I); or a salt, especially a pharmaceutically acceptable salt with a base, thereof or a lactone thereof wherein the element (a) represents —CH | 12-18-2008 |
| 20090111995 | Process for the manufacture valsartan - The present invention relates to a process for the manufacture of an angiotensin receptor blocker (ARB; also called angiotension II receptor antagonist or AT | 04-30-2009 |
| 20090137805 | N-PHENYL-2-PYRIMIDINE-AMINE DERIVATIVES - The present invention relates to novel amides and a process for preparing these amides. | 05-28-2009 |
| 20090143340 | Pyrocatechin Derivatives - Pyrocatechin derivatives of formula I | 06-04-2009 |
| 20090275758 | PROCESS FOR PHENYLACETIC ACID DERIVATIVES - A process for the production of a compound of Formula I, or a pharmaceutically acceptable salt thereof, or a pharmaceutically acceptable prodrug ester thereof, | 11-05-2009 |
| 20100113801 | Process for preparing 5-biphenyl-4-amino-2-methyl pentanoic acid - The present invention relates to pyrrolidin-2-ones according to the formula (1), or salts thereof, | 05-06-2010 |
| 20100130749 | METHODS - The invention related to a novel process, novel process steps and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially renin inhibitors, such as Aliskiren Inter alia the invention relates to a process for the manufacture of a compound of the formula I. | 05-27-2010 |
| 20100184991 | PREPARATION OF TERAZOLE DERIVATIVES - The invention relates to a process for the preparation of (S)-pyrrolidine-1H-tetrazole derivatives of formula | 07-22-2010 |
| 20100184998 | ORGANIC COMPOUNDS - The present invention relates to olefin metathesis processes for the manufacture of a compound of the formula (I) | 07-22-2010 |
| 20100249429 | PROCESS FOR THE MANUFACTURE OF VALSARTAN - The present invention relates to a process for the manufacture of an angiotensin receptor blocker (ARB; also called angiotension II receptor antagonist or AT | 09-30-2010 |
| 20100267965 | 3-Alkyl-5- (4-alkyl-5-oxo-tetrahydrofutran-2-yl) pyrrolidin-2-one Derivatives as Intermediates in the Synthesis of Renin Inhibitors - The invention related to a novel process, novel process steps and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially renin inhibitors, such as Aliskiren. Inter alia, the invention relates to a process for the manufacture of a compound of the formula II, | 10-21-2010 |
| 20100274027 | ORGANIC COMPOUNDS - The invention provides a novel process, novel process steps and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially renin inhibitors, such as Allskiren. Inter alia, the invention provides a process for the manufacture of a compound of the formula III, | 10-28-2010 |
| 20110015425 | PROCESS - The present invention relates to improved processes for the production of 2-amino-2-[2-(4-C | 01-20-2011 |
| 20110137044 | ALTERNATIVE SYNTHESIS OF RENIN INHIBITORS AND INTERMEDIATES THEREOF - The present invention relates to synthetic routes to prepare a compound of the formula | 06-09-2011 |
| 20110144352 | PROCESSES FOR THE PREPARATION OF 4-OXO-OCTAHYDRO-INDOLE-1-CARBOCYCLIC ACID METHYL ESTER AND DERIVATIVES THEREOF - The present invention relates to a process for the production of carbamic acid (2-chloroethyl)(3-oxocyclohexyl)-alkyl ester enantiomers and of 1-carbalkoxy-4-ketoperhydroindole enantiomers. | 06-16-2011 |
| 20110184187 | PROCESS FOR THE PREPARATION OF TETRAZOLE DERIVATIVES FROM ORGANO BORON AND ORGANO ALUMINIUM AZIDES - The present invention relates to a method for preparing substituted tetrazoles, compounds obtained according to this method, new reactants and new tetrazole derivatives. | 07-28-2011 |
| 20120142916 | PROCESS FOR PREPARING 5-BIPHENYL-4-AMINO-2-METHYL PENTANOIC ACID - The present invention relates to pyrrolidin-2-ones according to the formula (1), or salts thereof, | 06-07-2012 |
| 20120226039 | N-Phenyl-2-pyrimidine-amine Derivatives - The present invention relates to novel amides and a process for preparing these amides. | 09-06-2012 |
| 20120238761 | PROCESS FOR THE MANUFACTURE OF ORGANIC COMPOUNDS - The present invention relates to processes for the manufacture of an angiotensin receptor blocker (ARB; also called angiotension II receptor antagonist or AT | 09-20-2012 |
| 20120330026 | PROCESS FOR THE PREPARATION OF TETRAZOLE DERIVATIVES FROM ORGANO BORON AND ORGANO ALUMINIUM AZIDES - The present invention relates to a method for preparing substituted tetrazoles, compounds obtained according to this method, new reactants and new tetrazole derivatives. | 12-27-2012 |
| 20130289127 | AMINOALKANOL DERIVATIVES - Disclosed are compounds of formula I | 10-31-2013 |
| 20140094625 | Process - The present invention relates to improved processes for the production of 2-amino-2-[2-(4-C | 04-03-2014 |
| 20140249320 | Process for Preparing 5-biphenyl-4-amino-2-methyl Pentanoic Acid - The present invention relates to pyrrolidin-2-ones according to the formula (1), or salts thereof, | 09-04-2014 |
| 20150018552 | N-Phenyl-2-pyrimidine-amine Derivatives - The present invention relates to novel amides and a process for preparing these amides. | 01-15-2015 |
