Patent application number | Description | Published |
20090131506 | Oxindoles as Kinase Inhibitors - The present invention relates to oxindoles of the formula I, their use as protein kinase activators or inhibitors, a method for their manufacture, their use for the preparation of a medicament for the treatment of diseases and their use for the manufacture of a pharmaceutical composition. | 05-21-2009 |
20090163556 | GLYCINAMIDE DERIVATIVES AS RAF-KINASE INHBITORS - The present invention relates to glycinamide derivatives of formula I, | 06-25-2009 |
20090197882 | INDAZOLE DERIVATIVES FOR THE TREATMENT OF HSP90-INDUCED DISEASES - Novel indazole derivatives of the formula (I), in which R | 08-06-2009 |
20090253688 | Semicarbazide derivatives as kinase inhibitors - The present invention relates to semicarbazide derivatives of formula I, the use of the compounds of formula I as inhibitors of one or more kinases, the use of the compounds of formula I for the manufacture of a pharmaceutical composition and a method of treatment, comprising administering said pharmaceutical composition to a patient. | 10-08-2009 |
20090298885 | METHYLENE UREA DERIVATIVES - The present invention relates to methylene urea derivatives of formula (I), the use of the compounds of formula (I) as inhibitors of raf-kinase, the use of the compounds of formula (I) for the manufacture of a pharmaceutical composition and a method of treatment, comprising administering said pharmaceutical composition to a patient. | 12-03-2009 |
20090325974 | 1,5-DIPHENYLPYRAZOLES II AS HSP90 INHIBITORS - Novel 1,5-diphenylpyrazole derivatives of the formula (I) in which R | 12-31-2009 |
20100022540 | TRIAZOLE DERIVATIVES II - Novel triazole derivatives of the formula (I) in which R | 01-28-2010 |
20100113542 | TRIAZOLE DERIVATIVE AS AN HSP 90 INHIBITOR - 5-[4-(2-Methylphenyl)-3-hydroxy-4H-1,2,4-triazol-5-yl]-2,4-dihydroxy-N-methyl-N-butylbenzamide is an HSP90 inhibitor and can be used for the preparation of a medicament for the treatment of diseases in which the inhibition, regulation and/or modulation of HSP90 plays a role. | 05-06-2010 |
20100173923 | 4 (PYRROLOPYRIDINYL)PYRIMIDINYL-2-AMINE DERIVATIVES - Compounds of the formula I in which R | 07-08-2010 |
20100197757 | OXINDOLES AS KINASE INHIBITORS - The present invention relates to oxindoles of the formula I, their use as protein kinase activators or inhibitors, a method for their manufacture, their use for the preparation of a medicament for the treatment of diseases and their use for the manufacture of a pharmaceutical composition. | 08-05-2010 |
20100234324 | Quinazolinamide derivatives - Novel quinazolinamide derivatives of the formula (I), in which R | 09-16-2010 |
20100292262 | 4 (PYRROLO[2,3-C]PYRIDINE-3-YL)PYRIMIDIN-2-AMINE DERIVATIVES - Compounds of the formula (I), in which R | 11-18-2010 |
20110028485 | 1,5-DIPHENYLPYRAZOLES II AS HSP90 INHIBITORS - Novel 1,5-diphenylpyrazole derivatives of the formula (I) in which R | 02-03-2011 |
20110082140 | 6-(PYRROLOPYRIDINYL) PYRIMIDIN-2-YLAMINE DERIVATIVES AND THE USE THEREOF FOR THE TREATMENT OF CANCER AND AIDS. - Compounds of the formula (I), in which R | 04-07-2011 |
20110092527 | 4 (Pyrrolopyridinyl)pyrimidin-2-ylamine derivatives - Compounds of the formula (I), in which R | 04-21-2011 |
20110136830 | CHROMENONE DERIVATIVES - Novel compounds of the formula I | 06-09-2011 |
20110245225 | QUINAZOLINAMIDE DERIVATIVES - Novel quinazolinamide derivatives of the formula (I), in which R | 10-06-2011 |
20120238582 | QUINAZOLINE DERIVATIVES - Novel quinazolinamide derivatives of the formula (I), in which R | 09-20-2012 |
20120264999 | 4 (PYRROLOPYRIDINYL)PYRIMIDIN-2-YLAMINE DERIVATIVES - Compounds of the formula (I), in which R | 10-18-2012 |
20130158076 | Methylene Urea Derivatives - The present invention relates to methylene urea derivatives of formula (I), the use of the compounds of formula (I) as inhibitors of raf-kinase, the use of the compounds of formula (I) for the manufacture of a pharmaceutical composition and a method of treatment, comprising administering said pharmaceutical composition to a patient. | 06-20-2013 |
20130178443 | PHENYLQUINAZOLINE DERIVATIVES - Novel quinazolinamide derivatives of the formula (I), in which R1-R43 and X have the meanings indicated in claim | 07-11-2013 |
20130310391 | 7-AZAINDOLE DERIVATIVES - Compounds of the formula (I) in which R, R | 11-21-2013 |