| Class / Patent application number | Description | Number of patent applications / Date published |
|---|
| 548235000 | Plural double bonds between the ring members of the oxazole ring | 11 |
| 20080221336 | Pparalpha/Gamma Agonists and Processes of Preparing - This invention provides a method for preparing compounds having the structure [Formula (I)] wherein L is [Formula (A)] or [Formula (B)] in which R | 09-11-2008 |
| 20090093639 | Prodrugs of carbamate inhibitors of IMPDH - The present invention relates to novel compounds, methods of preparing these compounds, and pharmaceutical compositions comprising these compounds. These compounds are carbamate prodrugs that convert to active inhibitors of the IMPDH enzyme in vivo. The compounds and pharmaceutical compositions of this invention are particularly well suited for activation and subsequent inhibition of the IMPDH enzyme activity. Consequently, these prodrugs may be advantageously used as therapeutic agents for IMPDH mediated processes. This invention also relates to methods for inhibiting the activity of IMPDH using the compounds and compositions of this invention. | 04-09-2009 |
| 20090149657 | PROCESS FOR THE SYNTHESIS OF INTERMEDIATES OF CHLORAMPHENICOL OR ITS ANALOGUES - The present invention relates to the synthesis of antibacterial compounds such as Chloramphenicol and its analogues Thiamphenicol and Florfenicol and particularly to a new reaction for the preparation of the intermediate compound aminodiolphenylsulfone. This reaction permits the introduction of modified residues to obtain modified antibiotics with an improved stability towards the action of bacterial resistant determinants. In addition, higher purities may be also obtained due to an improved procedure requiring fewer purification steps. | 06-11-2009 |
| 20100041896 | Macrolide compound with bis-oxazoly - This patent mainly provides a new macrolide compound named FW-04-806, which contains bis-oxazoly in molecule. FW-04-806, a bis-oxazolyl macrolide compound extracted and separated from the ferment liquid of | 02-18-2010 |
| 20150065727 | THE NEW DERIVATIVES OF (Z)-1,2-DIPHENYLETHENE - The present invention relates to the new chemical compounds containing (Z)-1,2-diphenylethene moiety in the structures, particularly the new derivatives of cis-stilbene, the new derivatives of 4,5-diphenyl-1,3-oxazole, the new derivatives of 1-methyl-4,5-diphenyl-1H-imidazole and pharmaceutically acceptable salts thereof. The invention relates also to the application of aforementioned compounds as a microtubule-interfering agents (MIAs). The new derivatives, because of their potential antimitotic and antiangio-genic activity, can be used as ingredients in the preparations used in the treatment of cancer. | 03-05-2015 |
| 548236000 | Cyano or -C(=X)-, wherein X is chalcogen, attached directly or indirectly to the oxazole ring by nonionic bonding | 6 |
| 20090221835 | PROCESSES FOR PREPARING BIARYL UREAS AND ANALOGS THEREOF - The present invention relates to processes for preparing biaryl ureas derivatives and analogs thereof. The invention also provides compounds useful as intermediates in the processes of the present invention. The process is useful for preparing compounds that inhibit IMPDH. | 09-03-2009 |
| 20100016609 | METHODS FOR THE PREPARATION OF AZOLE COMPOUNDS - The present invention is directed to processes, compositions and methods associated with the preparation of azole derivatives of formula I: | 01-21-2010 |
| 20100249428 | PROCESS FOR THE PREPARATION OF PROPIONIC ACID DERIVATIVES - The invention relates to a process for the preparation of a compound of formula (I) | 09-30-2010 |
| 20110301355 | Amidine compounds and herbicides - Novel amidine compounds which may be active ingredients in herbicides that are reliably effective at a lesser dose and highly safe, and herbicides containing these compounds as active ingredients are provided. Amidine compounds represented by a formula (1′) | 12-08-2011 |
| 20130184468 | PROCESS FOR THE PREPARATION OF PROPIONIC ACID DERIVATIVES - The invention relates to a process for the preparation of a compound of formula (I) | 07-18-2013 |
| 20150025249 | PROCESS FOR THE PREPARATION OF PROPIONIC ACID DERIVATIVES - The invention relates to a process for the preparation of a compound of formula (I) | 01-22-2015 |
