| Class / Patent application number | Description | Number of patent applications / Date published |
|---|
| 546186000 | Plural piperidine rings | 16 |
| 546187000 | Additional hetero ring containing | 4 |
| 20090118513 | Chemical Compounds - The present invention provides a compound of a formula (I): | 05-07-2009 |
| 20100029946 | CRYSTALLINE FORM OF A BENZIMIDAZOLE-CARBOXAMIDE MEDICINAL COMPOUND - The invention provides crystalline forms of the novel benzimidazole-carboxamide 5-HT | 02-04-2010 |
| 20110306767 | N-Substituted-Heterocycloalkyloxybenzamide Compounds and Methods of Use - The present invention provides N-substituted-heterocycloalkyloxybenzamide compounds, as well as pharmaceutical compositions and methods of use. One embodiment of the invention is a compound having the structure | 12-15-2011 |
| 20160137629 | COMPOUNDS FOR BINDING TO THE PLATELET SPECIFIC GLYCOPROTEIN IIb/IIIa AND THEIR USE FOR IMAGING OF THROMBI - The present invention relates to novel fluorine containing compounds, methods for their preparation, the intermediates of the synthesis, their use as diagnostic agents, especially for imaging of thrombi. The invention relates to positron emission tomography (PET) agents and associated precursor reagents, and methods for producing such radiolaveled agents for imaging of thrombi in a mammalian body. More particularly, the invention relates to small nonpeptide, high-affinity, specific-binding glycoprotein 11b/IIIa antagonists for imaging of thrombi. | 05-19-2016 |
| 546188000 | Chalcogen attached directly to a ring carbon of a piperidine ring by nonionic bonding | 7 |
| 20080255362 | Cyclic amide derivative, and its production and use - The present invention provides a cyclic amide derivative useful as a drug for treating thrombosis, which is represented by the formula (I): | 10-16-2008 |
| 20100249421 | BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS - This invention provides compounds of formula I: | 09-30-2010 |
| 20100305327 | NITROXYL COMPOUND, AND POLYMERIZATION INHIBITOR AND POLYMERIZATION INHIBITOR COMPOSITION USING SAME - The following compound, inhibitor, and composition are provided: a compound having low volatility, high nitroxyl group concentration, and high polymerization inhibitory activity; a polymerization inhibitor using the compound; and a polymerization inhibitor composition using the compound. | 12-02-2010 |
| 20110319625 | BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS - This invention provides compounds of formula I: | 12-29-2011 |
| 20120016130 | PROCESS FOR PREPARING A BIPHENYL-2-YLCARBAMIC ACID - The invention provides a process of preparing an intermediate useful in the synthesis of biphenyl-2-ylcarbamic acid 1-(2-{[4-(4-carbamoylpiperidin-1-ylmethyl)benzoyl]methylamino}ethyl)piperidin-4-yl ester, and a process of preparing a crystalline freebase of the ester. | 01-19-2012 |
| 20140121378 | PROCESS FOR PREPARING A BIPHENYL-2-YLCARBAMIC ACID - The invention provides a process of preparing an intermediate useful in the synthesis of biphenyl-2-ylcarbamic acid 1-(2-{[4-(4-carbamoylpiperidin-1-ylmethyl)benzoyl]methylamino}ethyl)piperidin-4-yl ester, and a process of preparing a crystalline freebase of the ester. | 05-01-2014 |
| 20140323734 | Method for the Preparation of N-Oxyl Hindered Amine Inhibitors - The present disclosure provides a composition and method for the preparation of N-oxyl hindered amine esters by contacting a compound of Formula (I), wherein R | 10-30-2014 |
| 546189000 | Having -C(=X)-, wherein X is chalcogen, bonded directly to a piperidine ring | 4 |
| 20120130076 | Synthetic Multimerizing Agents - New compounds are disclosed for multimerizing immunophilins and proteins containing immunophilin or immunophilin-related domains. The compounds are of the formula | 05-24-2012 |
| 20140171649 | Methods and Compositions for the Synthesis of Multimerizing Agents - The invention features methods and compositions for the synthesis of multimerizing agents. An exemplary method for producing AP20187 may comprise: (a) coupling 2-N,Ndimethylaminomethyl-1,3-diaminopropane with AP20792 to produce the dimeric alcohol, AP20793; and (b) coupling the AP20793 so produced with API7362 to yield AP20187. In particular embodiments, the method further includes the step of producing API7362 by coupling API7360 with methyl-L-pipecolic acid, or a salt thereof. | 06-19-2014 |
| 20150148543 | Methods and Compositions for the Synthesis of Multimerizing Agents - The invention features methods and compositions for the synthesis of multimerizing agents. | 05-28-2015 |
| 20160031810 | BENZIDINE DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING BENZIDINE DERIVATIVE FOR TREATING LIVER DISEASE CAUSED BY HEPATITIS C VIRUS - The disclosed compounds have antiviral activity against C-type virus, an optical isomer thereof, a pharmaceutically acceptable salt thereof, a method for preparing the same, and a pharmaceutical composition containing the same as an active ingredient for preventing or treating liver disease caused by hepatitis C virus. The benzidine derivative according to the present invention has excellent antiviral activity against hepatitis C virus and exhibits excellent medicinal activity in the living body, and thus the pharmaceutical composition containing the same as an active ingredient can be useful as a pharmaceutical composition for preventing or treating liver disease, such as acute hepatitis C, chronic hepatitis C, cirrhosis, or hepatocellular carcinoma, caused by C-type virus. | 02-04-2016 |
| 546190000 | Having -C(=X)-, wherein X is chalcogen, attached indirectly to a piperdine ring by nonionic bonding | 1 |
| 20100160637 | METHOD FOR THE PRODUCTION OF 4-FORMYLAMINOPIPERIDINE DERIVATIVES - Method for producing 4-formylaminopiperidine derivatives of the formula (I) | 06-24-2010 |
