Class / Patent application number | Description | Number of patent applications / Date published |
544140000 | 1,2-Diazole ring (including hydrogenated) | 10 |
20100152443 | PYRAZOLE DERIVATIVE, INTERMEDIATE THEREFOR, PROCESSES FOR PRODUCING THESE, AND HERBICIDE CONTAINING THESE AS ACTIVE INGREDIENT - The present invention provides a pyrazole derivative of the general formula (1), | 06-17-2010 |
20120029192 | Pyrazole Derivatives - This invention relates to pyrazole derivatives of formula (I) | 02-02-2012 |
20120316336 | 4-[-2-[[5-METHYL-1-(2-NAPHTALENYL)-1H-PYRAZOL-3-YL]OXY]ETHYL]MORPHOLINE HYDROCHLORIDE POLYMORPHS AND SOLVATES - The present invention relates to polymorphs and solvates of the hydrochloride salt of 4-[2-[[5-methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine (P027), processes for their preparation, and to pharmaceutical compositions comprising them. | 12-13-2012 |
20130150575 | 4-[-2-[[5-METHYL-1-(2-NAPHTALENYL)-1H-PYRAZOL-3-YL]OXY]ETHYL]MORPHOLINE HYDROCHLORIDE AMORPHOUS SOLID FORMS - The present invention relates to solid forms having a low degree of crystallinity or substantially amorphous of the hydrochloride salt of 4-[2-[[5-methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine (P027) and processes for their preparation. | 06-13-2013 |
20130267704 | 1-BENZYL-3-HYDROXYMETHYLINDAZOLE DERIVATIVES AND USE THEREOF IN THE TREATMENT OF DISEASES BASED ON THE EXPRESSION OF MCP-1, CX3CR1 AND P40 - The present invention relates to novel 1-benzyl-3-hydroxymethylindazole derivatives according to formula (I) described in the claims, and to a pharmaceutical composition comprising them, together with a pharmaceutically acceptable vehicle. In addition, the present invention relates to the use of 1-benzyl-3-hydroxymethylindazole derivatives for the preparation of a pharmaceutical composition that is active in the treatment of diseases based on the expression of MCP-1, CX3CR1 and p40, and to their use in a method for treating or preventing diseases based on the expression of MCP-1, CX3CR1 and p40. | 10-10-2013 |
20140011997 | NEPRILYSIN INHIBITORS - In one aspect, the invention relates to compounds having the formula: | 01-09-2014 |
20140073783 | NEPRILYSIN INHIBITORS - In one aspect, the invention relates to compounds having the formula: | 03-13-2014 |
20140364603 | NEPRILYSIN INHIBITORS - In one aspect, the invention relates to compounds having the formula: | 12-11-2014 |
20150073141 | DIARYL AND ARYLHETEROARYL UREA DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE PROPHYLAXIS AND TREATMENT OF DISORDERS RELATED THERETO - The present invention relates to certain pyrazole derivatives of Formula (I) and pharmaceutical compositions thereof that modulate the activity of the 5-HT | 03-12-2015 |
20150133658 | NEPRILYSIN INHIBITORS - In one aspect, the invention relates to compounds having the formula: | 05-14-2015 |