Patent application number | Description | Published |
20090054427 | AMINOBENZYL-SUBSTITUTED CYCLIC SULFONES USEFUL AS BACE INHIBITORS - The invention relates to novel heterocyclic compounds of the formula | 02-26-2009 |
20090099207 | Cyclic sulfones useful as BACE inhibitors - The invention relates to novel heterocyclic compounds of the formula | 04-16-2009 |
20100056490 | Cyclic sulfones with aminobenzyl substitution useful as BACE inhibitors - The invention relates to novel heterocyclic compounds of the formula | 03-04-2010 |
20100144741 | ETHANOLAMINE DERIVATIVES USEFUL AS BACE INHIBITORS - The invention relates to novel cyclic compounds of the formula (I), in free base form or in acid addition salt form, to their preparation, to their use as medicaments and to medicaments comprising them. | 06-10-2010 |
20110021520 | OXAZINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS - The invention relates to novel heterocyclic compounds of the formula | 01-27-2011 |
20110137044 | ALTERNATIVE SYNTHESIS OF RENIN INHIBITORS AND INTERMEDIATES THEREOF - The present invention relates to synthetic routes to prepare a compound of the formula | 06-09-2011 |
20120172359 | Oxazine Derivatives and their Use in the Treatment of Neurological Disorders - The invention relates to novel heterocyclic compounds of the formula | 07-05-2012 |
20120184539 | Novel Heterocyclic Derivatives and Their Use in the Treatment of Neurological Disorders - The invention relates to novel heterocyclic compounds of the formula | 07-19-2012 |
20130172331 | NOVEL OXAZINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE - The invention relates to novel oxazine derivatives of formula (I), and pharmaceutically acceptable salts thereof, | 07-04-2013 |
20130225574 | OXAZOLIDIN-2-ONE COMPOUNDS AND USES THEREOF - The present invention relates to oxazolidin-2-one substituted pyrimidine compounds that act as PI3K (phosphatidylinositol-3-kinase) inhibitors, as well as pharmaceutical compositions thereof, methods for their manufacture and uses for the treatment of conditions, diseases and disorders dependent on PI3K. | 08-29-2013 |
20130281449 | Oxazine Derivatives and their Use in the Treatment of Neurological Disorders - The invention relates to novel heterocyclic compounds of the formula (I), in which all of the variables are as defined in the specification, in free form or in pharmaceutically acceptable salt form, to their preparation, to their medical use and to medicaments comprising them. | 10-24-2013 |
20140107118 | Novel Heterocyclic Derivatives and Their Use in the Treatment of Neurological Disorders - The invention relates to novel heterocyclic compounds of the formula | 04-17-2014 |
20140135330 | Oxazolidin-2-one-Pyrimidine Derivatives - The present invention relates to oxazolidin-2-one substituted pyrimidine compounds that act as PI3K (phosphatidylinositol-3-kinase) inhibitors, as well as pharmaceutical compositions thereof, methods for their manufacture and uses for the treatment of conditions, diseases and disorders dependent on PI3K. | 05-15-2014 |
20140256715 | Novel Oxazine Derivatives and their use in the Treatment of Disease - The invention relates to novel oxazine derivatives of formula (I), and pharmaceutically acceptable salts thereof, in which all of the variables are as defined in the specification, pharmaceutical compositions thereof, combinations thereof, and their use as medicaments, particularly for the treatment of Alzheimer's Disease or diabetes via inhibition of BACE-1 or BACE-2. | 09-11-2014 |
20140349990 | Pyrazolopyrrolidine Derivatives and their Use in the Treatment of Disease - The present invention provides a compound of formula (I) or a pharmaceutically acceptable salt thereof; | 11-27-2014 |
20140378450 | OXAZOLIDIN-2-ONE COMPOUNDS AND USES THEREOF - The present invention relates to oxazolidin-2-one substituted pyrimidine compounds that act as PI3K (phosphatidylinositol-3-kinase) inhibitors, as well as pharmaceutical compositions thereof, methods for their manufacture and uses for the treatment of conditions, diseases and disorders dependent on PI3K. | 12-25-2014 |